Cart
sales@molnova.com
Home - Products - GPCR/G Protein - Histamine Receptor - Pitolisant hydrochloride

Pitolisant hydrochloride

CAS No. 903576-44-3

Pitolisant hydrochloride ( Ciproxidine;BF 2649;BF2649;BF-2649 )

Catalog No. M16495 CAS No. 903576-44-3

A potent and selective antagonist of H3 receptor with Ki/EC50 of 0.16/1.5 nM.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
5MG 39 In Stock
10MG 61 In Stock
25MG 113 In Stock
50MG 186 In Stock
100MG 295 In Stock
200MG 443 In Stock
500MG 708 In Stock
1G Get Quote In Stock
Group Booking Get Quotation Bulk Inquiry Add to Cart

Biological Information

  • Product Name
    Pitolisant hydrochloride
  • Note
    Research use only, not for human use.
  • Brief Description
    A potent and selective antagonist of H3 receptor with Ki/EC50 of 0.16/1.5 nM.
  • Description
    A potent and selective antagonist of H3 receptor with Ki/EC50 of 0.16/1.5 nM; no effect on H1, H2, H4 receptors (IC50>10 uM); orally bioactive.Sleep Disorder Approved
  • Synonyms
    Ciproxidine;BF 2649;BF2649;BF-2649
  • Pathway
    GPCR/G Protein
  • Target
    Histamine Receptor
  • Recptor
    Histamine Receptor
  • Research Area
    Neurological Disease
  • Indication
    Sleep Disorder

Chemical Information

  • CAS Number
    903576-44-3
  • Formula Weight
    332.31
  • Molecular Formula
    C17H27Cl2NO
  • Purity
    >98% (HPLC)
  • Solubility
    DMSO: ≥ 43 mg/mL
  • SMILES
    C1CCN(CC1)CCCOCCCC2=CC=C(C=C2)Cl.Cl
  • Chemical Name
    Piperidine, 1-[3-[3-(4-chlorophenyl)propoxy]propyl]-, hydrochloride (1:1)

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1. Ligneau X, et al. J Pharmacol Exp Ther. 2007 Jan;320(1):365-75.
2. Dudek M, et al. Metab Brain Dis. 2016 Oct;31(5):1023-9.
3. Ligneau X, et al. Biochem Pharmacol. 2007 Apr 15;73(8):1215-24.
Calculator

Molecular Weight Calculator

Dilution Calculator

Molarity Calculator

molnova catalog
related products

  • Psoralenoside

    Psoralenoside is a natural product isolated from the fruits of Psoralea corylifolia, shows estrogen-like activity, osteoblastic proliferation accelerating activity, antitumor effects and antibacterial activity.

  • Betahistine dihydroc...

    Betahistine Dihydrochloride is a histamine H3 receptors inhibitor used as an antivertigo drug.

  • Orphenadrine hydroch...

    Orphenadrine is an anticholinergic drug of the ethanolamine antihistamine class with prominent central nervous system (CNS) and peripheral actions used to treat painful muscle spasms and other similar conditions, as well as the treatment of some aspects of Parkinson's disease.

Sign In Join Free